发明名称 METHOD FOR PREPARING 4-METHYLAMINO-4-PHENYLPIPERIDINE
摘要 The invention concerns a method for preparing a 4-alkoxycarbonylamino-1-benzyl-4-phenylpiperidine of formula (I) by hydrolysis of 1-benzyl-4-cyano-4-phenylpiperidine (II) in acid medium and treatment of 1-benzyl-4-phenyl-4-piperidinecarboxamide (III) thus obtained with bromine in the presence of an alkaline alcoholate. The invention also concerns a method for preparing 4-methylamino-4-phenylpiperidine from said compound (II).
申请公布号 WO03008381(A1) 申请公布日期 2003.01.30
申请号 WO2002FR02498 申请日期 2002.07.15
申请人 SANOFI-SYNTHELABO;ANNE-ARCHARD, GILLES;GROS-CLAUDE, PATRICK 发明人 ANNE-ARCHARD, GILLES;GROS-CLAUDE, PATRICK
分类号 C07D211/58;(IPC1-7):C07D211/58 主分类号 C07D211/58
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