发明名称 CYCLIC AMINO ACID DERIVATIVES
摘要 Novel compounds of formula (I), wherein R1, R2, R2', R2'', R3, R4, R5, R5', R5'', R5''', R5'''', X, Y, U, V and W have the meanings given in claim no.1, are inhibitors of the coagulation factors Xa and VIIa and can be used for treating thromboses, myocardial infarct, arteriosclerosis, infections, apoplexia, angina pectoris, restenosis following angioplasty, intermittent claudication, tumors, tumor diseases and/or tumor metastases.
申请公布号 CA2415964(A1) 申请公布日期 2003.01.17
申请号 CA20012415964 申请日期 2001.07.03
申请人 MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG 发明人 GLEITZ, JOHANNES;BARNES, CHRISTOPHER;JURASZYK, HORST;DORSCH, DIETER;TSAKLAKIDIS, CHRISTOS;MEDERSKI, WERNER
分类号 C07D295/20;A61K31/397;A61K31/402;A61K31/4166;A61K31/421;A61K31/426;A61K31/4439;A61K31/451;A61K31/495;A61K45/00;A61P7/02;A61P7/04;A61P9/00;A61P9/10;A61P25/00;A61P29/00;A61P35/00;A61P43/00;C07D205/04;C07D207/16;C07D207/28;C07D211/34;C07D211/60;C07D233/34;C07D233/36;C07D263/06;C07D263/24;C07D277/06;C07D401/04;C07D413/12;(IPC1-7):C07D401/04;C07D233/02;C07D241/04;C07D207/08;A61K31/40 主分类号 C07D295/20
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