发明名称 KINETIC RESOLUTION OF A INTERMEDIATE USEFUL IN THE PRODUCTION OF BENAZEPRIL AND ANALOGUES THEREOF
摘要 The present invention provides an efficient synthetic process for making benazepril and analogues thereof by having an intermediate compound undergo epimerization and kinetic resolution.
申请公布号 WO03003972(A2) 申请公布日期 2003.01.16
申请号 WO2002IB03060 申请日期 2002.05.20
申请人 SCINOPHARM TAIWAN, LTD.;TSENG, WEI-HONG;SCHLOEMER, GEORGE;CHENG, KAU, MING;CHEN, CHIEN, WEN;CHENG, CHIH, WEN 发明人 TSENG, WEI-HONG;SCHLOEMER, GEORGE;CHENG, KAU, MING;CHEN, CHIEN, WEN;CHENG, CHIH, WEN
分类号 A61K31/55;A61P9/02;A61P9/12;A61P13/12;A61P43/00;C07B53/00;C07B55/00;C07B61/00;C07D223/16 主分类号 A61K31/55
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