发明名称 AMINOALCOHOL DERIVATIVES
摘要 <p>A compound of the formula (I) wherein X1 is bond or -O(CH2)m- (in which m is an integral number of 1, 2 or 3); X2 is bond, -(CH2)n-, etc. (in which n is an integral number of 1, 2 or 3); R1 is hydrogen or amino protective group; R2 is hydroxy(lower)alkyl or (lower)alkoxy(lower)alkyl; A is phenyl, pyridyl, indolyl or carbazolyl, each of which may be substituted with one or two substituent(s) selected from the group consisting of halogen, hydroxy, lower alkyl, etc.; and B is phenyl or pyridyl, each of which may be substituted with one or two substituent(s) selected from the group consisting of halogen, hydroxy, nitro, etc.; and a pharmaceutically acceptable salt thereof which is useful as a medicament.</p>
申请公布号 WO0162705(A3) 申请公布日期 2003.01.16
申请号 WO2001JP01442 申请日期 2001.02.26
申请人 FUJISAWA PHARMACEUTICAL CO., LTD.;TANIGUCHI, KIYOSHI;KAYAKIRI, HIROSHI;SAKURAI, MINORU;FUJII, NAOAKI;WASHIZUKA, KENICHI;HAMASHIMA, HITOSHI;TOMISHIMA, YASUYO;HAMADA, KAORI;YAMAMOTO, NOBUHIRO;ISHIKAWA, HIROFUMI;UNAMI, NAOKO;MIURA, TOSHIKO 发明人 TANIGUCHI, KIYOSHI;KAYAKIRI, HIROSHI;SAKURAI, MINORU;FUJII, NAOAKI;WASHIZUKA, KENICHI;HAMASHIMA, HITOSHI;TOMISHIMA, YASUYO;HAMADA, KAORI;YAMAMOTO, NOBUHIRO;ISHIKAWA, HIROFUMI;UNAMI, NAOKO;MIURA, TOSHIKO
分类号 A61K31/195;A61K31/403;A61K31/4045;A61K31/4406;A61K31/4439;A61P1/04;A61P1/16;A61P1/18;A61P3/00;A61P3/04;A61P3/06;A61P3/10;A61P9/10;A61P9/12;A61P11/04;A61P13/02;A61P13/04;A61P25/24;A61P27/06;A61P43/00;C07C213/04;C07C217/30;C07C217/32;C07C217/34;C07C217/70;C07C217/86;C07C225/16;C07C229/34;C07C229/38;C07C237/30;C07C271/28;C07C311/08;C07C311/17;C07C311/21;C07C311/40;C07D209/08;C07D209/14;C07D209/88;C07D213/65;C07D401/12;(IPC1-7):C07C217/86;C07D471/04;C07C311/18;A61K31/133 主分类号 A61K31/195
代理机构 代理人
主权项
地址