发明名称 AZAINDOLES
摘要 The invention is directed to physiologically active compounds of general formula (I): and compositions containing such compounds; and their prodrugs, and pharmaceutically acceptable salts and solvates of such compounds and their prodrugs, as well as to novel compounds within the scope of formula (I). Such compounds and compositions have valuable pharmaceutical properties, in particular the ability to inhibit kinases.
申请公布号 WO03000688(A1) 申请公布日期 2003.01.03
申请号 WO2002GB02799 申请日期 2002.06.20
申请人 AVENTIS PHARMA LIMITED;COX, PAUL, JOSEPH;MAJID, TAHIR, NADEEM;LAI, JUSTINE, YEUN, QUAI;MORLEY, ANDREW;AMENDOLA, SHELLEY;DEPRETS, STEPHANIE, DANIELE;EDLIN, CHRIS;GARDNER, CHARLES, J.;KOMINOS, DOROTHEA;PEDGRIFT, BRIAN, LESLIE;HALLEY, FRANK;GILLESPY, TIMOTHY, ALAN;EDWARDS, MICHAEL;CLERC, FRANCOIS, FREDERIC;NEMECEK, CONCEPTION;HOUILLE, OLIVIER;DAMOUR, DOMINIQUE;BOUCHARD, HERVE;BEZARD, DANIEL;CARREZ, CHANTAL 发明人 COX, PAUL, JOSEPH;MAJID, TAHIR, NADEEM;LAI, JUSTINE, YEUN, QUAI;MORLEY, ANDREW;AMENDOLA, SHELLEY;DEPRETS, STEPHANIE, DANIELE;EDLIN, CHRIS;GARDNER, CHARLES, J.;KOMINOS, DOROTHEA;PEDGRIFT, BRIAN, LESLIE;HALLEY, FRANK;GILLESPY, TIMOTHY, ALAN;EDWARDS, MICHAEL;CLERC, FRANCOIS, FREDERIC;NEMECEK, CONCEPTION;HOUILLE, OLIVIER;DAMOUR, DOMINIQUE;BOUCHARD, HERVE;BEZARD, DANIEL;CARREZ, CHANTAL
分类号 A61K;A61K31/437;A61K31/4709;A61K31/4725;A61K31/496;A61K31/4985;A61K31/5355;A61K31/5377;A61K31/541;A61P;A61P9/00;A61P11/00;A61P11/02;A61P11/06;A61P13/08;A61P17/00;A61P17/02;A61P17/06;A61P19/02;A61P27/14;A61P29/00;A61P35/00;A61P37/08;A61P43/00;C07D;C07D471/04;C07D487/04;C07D519/00;(IPC1-7):C07D471/04;A61K31/498 主分类号 A61K
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