发明名称 |
GLUCOPYRANOSYLOXY BENZYLBENZENE DERIVATIVES, MEDICINAL COMPOSITIONS CONTAINING THE SAME AND INTERMEDIATES FOR THE PREPARATION OF THE DERIVATIVES |
摘要 |
<p>The present invention relates to glucopyranosyloxybenzylbenzene derivatives represented by the general formula: <CHEM> wherein R<1> represents a hydrogen atom or a hydroxy( lower alkyl) group; and R<2> represents a lower alkyl group, a lower alkoxy group, a lower alkylthio group, a hydroxy(lower alkyl) group, a hydroxy(lower alkoxy) group, a hydroxy(lower alkylthio) group etc., and salts thereof, which have an excellent inhibitory activity in human SGLT2 and are useful as agents for the prevention or treatment of diabetes, obesity etc., and intermediates thereof.</p> |
申请公布号 |
EP1270584(A1) |
申请公布日期 |
2003.01.02 |
申请号 |
EP20010912380 |
申请日期 |
2001.03.15 |
申请人 |
KISSEI PHARMACEUTICAL CO., LTD. |
发明人 |
FUJIKURA, HIDEKI;FUSHIMI, NOBUHIKO;NISHIMURA, TOSHIHIRO;TATANI, KAZUYA;KATSUNO, KENJI;HIRATOCHI, MASAHIRO;TOKUTAKE, YOSHIKI;ISAJI, MASAYUKI |
分类号 |
A61P43/00;A61K31/7034;A61P3/04;A61P3/10;C07C39/04;C07C69/16;C07C69/18;C07C69/78;C07C323/18;C07H15/203;(IPC1-7):C07H15/203;C07C43/23;A61K31/703;C07C39/15 |
主分类号 |
A61P43/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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