发明名称 |
Crystalline forms of 1S-[1alpha(2S*,3R*), 9ALPHA]-6, 10-dioxo-N(2-ethoxy-5-oxo-tetrahydro-3-furanyl) -9-[[(1-isoquinolyl) carbonyl]-amino] octahydro-6H-piridazino[1,2-A][1,2] diazepin- 1-carboxamide |
摘要 |
A crystalline form of anhydrous 1S-[1alpha(2S*,3R*), 9ALPHA]-6, 10-dioxo-N(2-ethoxy-5-oxo-tetrahydro-3-furanyl)-9-[[(1-isoquinolyl) carbonyl]-amino] octahydro-6H-piridazino[1,2-A][1,2] diazepin-1-carboxamide which doesn't have the drawbacks of the currently known amorphous form of said compound; and a process for its preparation.
|
申请公布号 |
NZ507199(A) |
申请公布日期 |
2002.12.20 |
申请号 |
NZ19990507199 |
申请日期 |
1999.04.07 |
申请人 |
HOECHST MARION ROUSSEL |
发明人 |
GODARD, JEAN-YVES;ROGNON, VALERIE |
分类号 |
C07D487/04;A61K31/551;A61K38/00;A61K38/06;A61P25/00;A61P29/00;A61P37/00;A61P37/02;A61P43/00;C07K5/02;C07K5/023;(IPC1-7):C07K5/023;A61K31/55 |
主分类号 |
C07D487/04 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|