发明名称 Crystalline forms of 1S-[1alpha(2S*,3R*), 9ALPHA]-6, 10-dioxo-N(2-ethoxy-5-oxo-tetrahydro-3-furanyl) -9-[[(1-isoquinolyl) carbonyl]-amino] octahydro-6H-piridazino[1,2-A][1,2] diazepin- 1-carboxamide
摘要 A crystalline form of anhydrous 1S-[1alpha(2S*,3R*), 9ALPHA]-6, 10-dioxo-N(2-ethoxy-5-oxo-tetrahydro-3-furanyl)-9-[[(1-isoquinolyl) carbonyl]-amino] octahydro-6H-piridazino[1,2-A][1,2] diazepin-1-carboxamide which doesn't have the drawbacks of the currently known amorphous form of said compound; and a process for its preparation.
申请公布号 NZ507199(A) 申请公布日期 2002.12.20
申请号 NZ19990507199 申请日期 1999.04.07
申请人 HOECHST MARION ROUSSEL 发明人 GODARD, JEAN-YVES;ROGNON, VALERIE
分类号 C07D487/04;A61K31/551;A61K38/00;A61K38/06;A61P25/00;A61P29/00;A61P37/00;A61P37/02;A61P43/00;C07K5/02;C07K5/023;(IPC1-7):C07K5/023;A61K31/55 主分类号 C07D487/04
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