发明名称 PROCESSO PARA A PREPARACAO DE DERIVADOS DE ACIDO AZABICICLO-NAFTIRIDINOCARBOXILICO COMPREENDENDO UM DIPEPTIDEO
摘要 <p>PCT No. PCT/IB96/00257 Sec. 371 Date Mar. 11, 1998 Sec. 102(e) Date Mar. 11, 1998 PCT Filed Mar. 27, 1996 PCT Pub. No. WO97/00268 PCT Pub. Date Jan. 3, 1997A multi-step process for preparing a dipeptide derivative of 7-(6-amino-3-azabicyclo[3.1.0.]hex-3-yl)-6-fluoro-1-(2,4-difluorophenyl)-1,4-dihydro-4-oxo-1,8-naphthyridine-3-carboxylic acid, in the form of a pharmaceutically acceptable acid addition salt is disclosed.</p>
申请公布号 PT833837(E) 申请公布日期 2002.11.29
申请号 PT19960904996T 申请日期 1996.03.27
申请人 PFIZER INC. 发明人 HARRY A. WATSON, JR.;TAMIM F. BRAISH;MICHAEL J. CASTALDI
分类号 C07D471/04;A61K31/435;A61P43/00;C07K1/06;C07K5/06;C07K5/062;(IPC1-7):C07K1/06;A61K31/47 主分类号 C07D471/04
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