发明名称 TRISUBSTITUTED-N-[(1S)-1,2,3,4-TETRAHYDRO-1-NAPHTHALENYL] BENZAMIDES WHICH INHIBIT P2X3 AND P2X2/3 CONTAINING RECEPTORS
摘要 Compounds of formula (I), are novel P2X>3< and P2X>2</P2X>3< antagonists which are useful in treating pain, urinary incontinence and bladder overactivity.
申请公布号 WO02094767(A2) 申请公布日期 2002.11.28
申请号 WO2002US15174 申请日期 2002.05.14
申请人 ABBOTT LABORATORIES 发明人 LEE, CHIH-HUNG;PERNER, RICHARD, J.;LARSON, DANIEL, P.;KOENIG, JOHN, R.;GOMTSYAN, ARTHUR, R.;ZHENG, GUO ZHU;DIDOMENICO, STANLEY;STEWART, ANDREW, O.;BAYBURT, EROL, K.
分类号 A61K31/194;A61K31/275;A61K31/277;A61K31/351;A61K31/381;A61K31/40;A61K31/4402;A61K31/4406;A61K31/505;A61P13/00;A61P13/02;A61P13/10;A61P21/00;A61P25/04;A61P43/00;C07C233/65;C07C233/66;C07C233/74;C07C233/76;C07C233/79;C07C251/48;C07C251/52;C07C255/60;C07C311/51;C07C321/24;C07D207/06;C07D213/40;C07D213/68;C07D213/71;C07D239/34;C07D309/12;C07D309/32;C07D317/72;C07D333/20;C07D333/34;C07D333/40;C07D333/42;C07D333/68;C07D333/72 主分类号 A61K31/194
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