发明名称 NOVEL PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS
摘要 Novel pyrrazole derivative compounds and their use as pharmaceutical agents, in particular their use as TGF-beta signal transduction inhibitors. The disclosed invention relates to compounds of the structure (I) wherein (I) is a four, five, or six membered saturated ring and X is C, O or S.
申请公布号 CA2446820(A1) 申请公布日期 2002.11.28
申请号 CA20022446820 申请日期 2002.05.13
申请人 ELI LILLY AND COMPANY 发明人 MILLER, SHAWN CHRISTOPHER;GOODSON, THEODORE JR.;GODFREY, ALEXANDER GLENN;SMITH, EDWARD C. R.;HERRON, DAVID KENT;MORT, NICOLAS ANTHONY;MCMILLEN, WILLIAM THOMAS;YINGLING, JONATHAN MICHAEL;DECOLLO, TODD VINCENT;CIAPETTI, PAOLA;SAWYER, JASON SCOTT;LI, HONG-YU;LIAO, JUNKAI;BEIGHT, DOUGLAS WADE
分类号 A61K31/4439;A61K31/444;A61K31/4709;A61K31/496;A61K31/5383;A61K31/55;A61K45/00;A61P3/10;A61P7/04;A61P9/10;A61P13/12;A61P17/02;A61P17/12;A61P19/02;A61P21/02;A61P25/28;A61P27/02;A61P29/00;A61P31/00;A61P31/18;A61P35/00;A61P37/02;A61P37/08;A61P43/00;C07D401/12;C07D471/04;C07D487/04;C07D498/04;(IPC1-7):C07D487/04;A61K31/33;A61K31/41;A61K31/535 主分类号 A61K31/4439
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