发明名称 METHOD FOR PRODUCING SULFONE DERIVATIVE
摘要 PROBLEM TO BE SOLVED: To provide a method for producing a sulfone derivative. SOLUTION: This method for producing the sulfone derivative represented by the general formula: R-W-S(O)2 -X-Y-L<2> (IIIa) (wherein, R is a cyclic hydrocarbon which may be substituted or the like; W is a bond or a divalent chain hydrocarbon group which may be substituted; X is a divalent chain hydrocarbon group which may be substituted; Y is -N(R<5> )-,-CO-, -S(O)-, -S(O)2 -, -CH2 - or a bond; L<2> is a hydrogen atom, a hydroxy group or an alkoxy group which may be substituted; and R<5> is a hydrogen atom or the like) or a salt thereof is characterized in that a sulfinic acid derivative represented by the general formula: R-W-S(O)2 -M (I) (wherein, M is a hydrogen atom, an alkali metal or an alkaline earth metal; R and W have the same meanings as the above- mentioned) with a compound represented by the formula; L<1> -X-Y-L<2> (IIa) (wherein, L<1> is a leaving group; and X, Y and L<2> have the same meanings as the above-mentioned).
申请公布号 JP2002338565(A) 申请公布日期 2002.11.27
申请号 JP20020070442 申请日期 2002.03.14
申请人 TAKEDA CHEM IND LTD 发明人 MIZUFUNE HIDEYA;YAMAMOTO HIROAKI;MIKI MASATAKA
分类号 C07D401/04;C07C315/04;C07C317/44;(IPC1-7):C07D401/04 主分类号 C07D401/04
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