发明名称 Process for preparing 5-[2-ethoxy-5-(4-methylpiperazin-1-yl sulfonyl)phenyl]-1-methyl-3-n-propyl-1,6-dihydro-7H-pyrazolo[4,3-d]-pyrimidin-7-one and intermediates for this preparation process
摘要 <p>Zp sob v²roby 5-[2-ethoxy-5-(4-methylpiperazin-1-ylsulfonyl)fenyl]-1-methyl-3-n-propyl-1,6-dihydro-7H-pyrazolo[4,3-d]pyrimidin-7-onu vzorce I, p°i n m se cyklizuje slou enina vzorce II, za bazick²ch, neutr ln ch nebo kysel²ch podm nek. Meziprodukty pro tento zp sob vzorce II a V./</p>
申请公布号 CZ290942(B6) 申请公布日期 2002.11.13
申请号 CZ19970001811 申请日期 1997.06.12
申请人 PFIZER RESEARCH AND DEVELOPMENT COMPANY, N. V./S. 发明人 DUNN PETER JAMES;WOOD ALBERT SHAW
分类号 C07D295/22;A61K31/00;A61K31/505;A61K31/519;A61K31/635;A61P13/02;A61P15/00;A61P15/10;C07B61/00;C07D;C07D231/14;C07D231/40;C07D295/26;C07D403/12;C07D487/04;(IPC1-7):C07D487/04 主分类号 C07D295/22
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