发明名称 |
Process for preparing 5-[2-ethoxy-5-(4-methylpiperazin-1-yl sulfonyl)phenyl]-1-methyl-3-n-propyl-1,6-dihydro-7H-pyrazolo[4,3-d]-pyrimidin-7-one and intermediates for this preparation process |
摘要 |
<p>Zp sob v²roby 5-[2-ethoxy-5-(4-methylpiperazin-1-ylsulfonyl)fenyl]-1-methyl-3-n-propyl-1,6-dihydro-7H-pyrazolo[4,3-d]pyrimidin-7-onu vzorce I, p°i n m se cyklizuje slou enina vzorce II, za bazick²ch, neutr ln ch nebo kysel²ch podm nek. Meziprodukty pro tento zp sob vzorce II a V./</p> |
申请公布号 |
CZ290942(B6) |
申请公布日期 |
2002.11.13 |
申请号 |
CZ19970001811 |
申请日期 |
1997.06.12 |
申请人 |
PFIZER RESEARCH AND DEVELOPMENT COMPANY, N. V./S. |
发明人 |
DUNN PETER JAMES;WOOD ALBERT SHAW |
分类号 |
C07D295/22;A61K31/00;A61K31/505;A61K31/519;A61K31/635;A61P13/02;A61P15/00;A61P15/10;C07B61/00;C07D;C07D231/14;C07D231/40;C07D295/26;C07D403/12;C07D487/04;(IPC1-7):C07D487/04 |
主分类号 |
C07D295/22 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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