发明名称 STABLE EMULSION COMPOSITIONS
摘要 <p>An emulsion composition containing a compound represented by the formula: <CHEM> wherein R is an aliphatic hydrocarbon group optionally having substituents, an aromatic hydrocarbon group optionally having substituents, a heterocyclic group optionally having substituents, a group represented by the formula: -OR<1> (wherein R<1> is a hydrogen atom or an aliphatic hydrocarbon group optionally having substituents) or a group represented by the formula: <CHEM> wherein R<1b> is a hydrogen atom or an aliphatic hydrocarbon group optionally having substituents, R<1c> is the same as or different from R<1b> and is a hydrogen atom or an aliphatic hydrocarbon group optionally having substituents, R<0> is a hydrogen atom or an aliphatic hydrocarbon group, or R and R<0> in combination represent a bond, Ar is an aromatic hydrocarbon group optionally having substituents <CHEM> or <CHEM> and the like, and n is an integer of 1 to 4, a salt thereof or a prodrug thereof, wherein the composition is adjusted to have a pH of not more than about 6, shows improved stability of the compound, a salt thereof or a prodrug thereof, and realizes expression of superior efficacy.</p>
申请公布号 EP1254659(A1) 申请公布日期 2002.11.06
申请号 EP20010948912 申请日期 2001.02.01
申请人 TAKEDA PHARMACEUTICAL COMPANY LIMITED 发明人 SATO, JUN
分类号 A61K9/107;A61K31/215;A61K31/235;A61K31/27;A61K31/41;A61K31/4192;A61K31/4196;A61K31/428;A61K47/10;A61K47/24;A61K47/44;A61P9/00;A61P25/00;A61P29/00;A61P31/00;A61P37/06;C07C311/14;C07D275/06;(IPC1-7):A61K31/215;A61K9/10 主分类号 A61K9/107
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