发明名称 N-Piperidino-5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-ethylpyrazole-3-carboxamide
摘要 <p>N-piperidino-5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-ethylpyrazole- 3-carboxamide of formula I, its salts and solvates. A process for preparing these compounds characterized in that a functional derivative of 5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-ethylpyrazole-3-carboxylic acid of formula II is reacted with 1-aminopiperidine with subsequent optional conversion to one of its salts or solvates. These compounds are used for treating disease involving the cannabinoid CB1 receptors.</p>
申请公布号 NZ512886(A) 申请公布日期 2002.10.25
申请号 NZ20000512886 申请日期 2000.01.28
申请人 SANOFI-SYNTHELABO 发明人 CAMUS, PHILIPPE;MARTINEZ, SERGE;RINALDI, MURIELLE;BARTH, FRANCIS
分类号 A61K31/415;A61K31/454;A61P3/00;A61P3/04;A61P25/00;A61P25/18;A61P25/28;A61P25/32;A61P25/34;A61P43/00;C07C69/738;C07C251/80;C07D231/14;(IPC1-7):C07D231/14;C07D401/12 主分类号 A61K31/415
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