发明名称 Indolylpiperidine derivatives as antihistaminic and antiallergic agents
摘要 Indolylpiperidine compounds of formula (I) wherein: A1 represents an alkylene, alkyleneoxy, alkylenethio, alkanoyl or hydroxyalkylene group; A2 represents a single bond, an alkylene or alkenylene group; W represents a single bond or a phenylene or furanylene group which is unsubstituted or substituted by one or more halogen atoms, alkoxy groups and/or alkyl groups; R1 represents a hydrogen atom or an alkyl, alkenyl, alkynyl, alkoxyalkyl, alkenyloxyalkyl, alkynyloxyalkyl alkoxy-alkoxyalkyl, phenylalkyl group wherein the phenyl ring is unsubstituted or substituted by one or more halogen atoms or alkyl, alkoxy or arylalkoxy groups, or a cycloalkylalkyl group wherein the cycloalkyl group is unsubstituted or substituted by one or more halogen atoms, alkyl groups or alkoxy groups; R2 represents a hydrogen or halogen atom or an alkyl or alkoxy group; and R3 represents a carboxyl group or a tetrazolyl group; and pharmaceutically acceptable salts thereof, process for their preparation and medicinal use
申请公布号 US2002147344(A1) 申请公布日期 2002.10.10
申请号 US20010006416 申请日期 2001.12.04
申请人 PAGES SANTACANA LLUIS;FONQUERNA POU SILVIA;PUIG DURAN CARLES;FERNANDEZ FORNER DOLORS 发明人 PAGES SANTACANA LLUIS;FONQUERNA POU SILVIA;PUIG DURAN CARLES;FERNANDEZ FORNER DOLORS
分类号 A61K31/445;A61K31/4525;A61K31/454;A61P11/02;A61P11/04;A61P11/06;A61P27/02;A61P37/08;C07D401/04;C07D401/14;C07D405/14;(IPC1-7):C0741/14;C0741/04 主分类号 A61K31/445
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