发明名称 TIOTROPIUM-CONTAINING INHALATION POWDER, A CAPSULE CONTAINING THE SAME AND THE USE THEREOF
摘要 Inhalation powder comprises a tiotropium salt (I) in admixture with excipients comprising coarse particles and fine particles. Inhalation powder comprises 0.04-0.8% of a tiotropium salt (I) in admixture with excipients comprising 80-99% coarse particles (average particle size 15-80 mum) and 1-20% fine particles (average particle size 1-9 mum). An Independent claim is also included for a capsule (inhalette) containing 3-10 mg of the inhalation powder.
申请公布号 SK7062002(A3) 申请公布日期 2002.10.08
申请号 SK20020000706 申请日期 2001.09.28
申请人 BOEHRINGER INGELHEIM PHARMA KG 发明人 BECHTOLD-PETERS KAROLINE;WALZ MICHAEL;BOECK GEORG;DOERR ROLF
分类号 C07D451/12;A61K9/00;A61K9/14;A61K9/51;A61K9/72;A61K31/439;A61K31/46;A61K47/02;A61K47/26;A61P11/00;A61P11/06;A61P43/00 主分类号 C07D451/12
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