发明名称 DIOXOLANE ANALOGS FOR IMPROVED INTER-CELLULAR DELIVERY
摘要 Compounds having the following formula:wherein: R1 is for example, H;C1-24 alkyl;C2-24 alkenyl;C6-24aryl;C5-20 heteroaromatic ring; orC3-20 non aromatic ring; R2 is a purine of pyrimidine group; or a pharmaceutically acceptable salt thereof, are useful in treating a patient having cancer.
申请公布号 WO0230922(A3) 申请公布日期 2002.09.26
申请号 WO2001CA01464 申请日期 2001.10.15
申请人 SHIRE BIOCHEM INC.;ATTARDO, GIORGIO;ZACHARIE, BOULOS;REJ, RABINDRA;LAVALLEE, JEAN-FRANCOIS;VAILLANCOURT, LOUIS;DENIS, REAL;LEVESQUE, SOPHIE 发明人 ATTARDO, GIORGIO
分类号 A61K31/513;A61K31/675;A61K31/7068;A61K38/00;A61P35/00;A61P35/02;A61P43/00;C07D405/04;C07D405/14;C07D473/18;C07F9/655;C07F9/6558;C07F9/6561;C07K5/06;C07K5/08;C07K5/10;C07K7/06 主分类号 A61K31/513
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