发明名称 |
DIOXOLANE ANALOGS FOR IMPROVED INTER-CELLULAR DELIVERY |
摘要 |
Compounds having the following formula:wherein: R1 is for example, H;C1-24 alkyl;C2-24 alkenyl;C6-24aryl;C5-20 heteroaromatic ring; orC3-20 non aromatic ring; R2 is a purine of pyrimidine group; or a pharmaceutically acceptable salt thereof, are useful in treating a patient having cancer. |
申请公布号 |
WO0230922(A3) |
申请公布日期 |
2002.09.26 |
申请号 |
WO2001CA01464 |
申请日期 |
2001.10.15 |
申请人 |
SHIRE BIOCHEM INC.;ATTARDO, GIORGIO;ZACHARIE, BOULOS;REJ, RABINDRA;LAVALLEE, JEAN-FRANCOIS;VAILLANCOURT, LOUIS;DENIS, REAL;LEVESQUE, SOPHIE |
发明人 |
ATTARDO, GIORGIO |
分类号 |
A61K31/513;A61K31/675;A61K31/7068;A61K38/00;A61P35/00;A61P35/02;A61P43/00;C07D405/04;C07D405/14;C07D473/18;C07F9/655;C07F9/6558;C07F9/6561;C07K5/06;C07K5/08;C07K5/10;C07K7/06 |
主分类号 |
A61K31/513 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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