发明名称 SUBSTITUTED BENZOINDOLES AS SPLA2 INHIBITORS
摘要 A novel class of benz[f]indole compounds see structure (I) is disclosed together with the use of such compounds for inhibiting sPLA2 mediated release of fatty acids for treatment of inflammatory diseases such as septic shock.
申请公布号 WO0250028(A3) 申请公布日期 2002.09.19
申请号 WO2001US43184 申请日期 2001.12.06
申请人 ELI LILLY AND COMPANY;BEIGHT, DOUGLAS, WADE;KINNICK, MICHAEL, DEAN;LIN, HO-SHEN;MORIN, JOHN, MICHAEL, JUNIOR;RICHETT, MICHAEL, ENRICO;SALL, DANIEL, JON;SAWYER, JASON, SCOTT;SMITH, EDWARD, C R 发明人 BEIGHT, DOUGLAS, WADE;KINNICK, MICHAEL, DEAN;LIN, HO-SHEN;MORIN, JOHN, MICHAEL, JUNIOR;RICHETT, MICHAEL, ENRICO;SALL, DANIEL, JON;SAWYER, JASON, SCOTT;SMITH, EDWARD, C R
分类号 A61K31/403;A61P1/04;A61P3/00;A61P3/12;A61P5/06;A61P5/18;A61P7/00;A61P7/04;A61P9/00;A61P11/00;A61P11/02;A61P11/06;A61P13/12;A61P17/02;A61P17/06;A61P19/02;A61P19/04;A61P19/06;A61P19/08;A61P21/00;A61P29/00;A61P31/04;A61P31/06;A61P31/10;A61P31/12;A61P35/00;A61P37/08;A61P43/00;C07D209/60 主分类号 A61K31/403
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