发明名称 SUBSTITUTED 8-ARYLQUINOLINE PHOSPHODIESTERASE-4 INHIBITORS
摘要 Novel sulfuric acid, methanesulfonic acid, p-toluenesulfonic acid, 2-naphthalenesulfonic acid, hydrochloride acid, or benzenesulfonic acid salts of substituted 8-arylquinolines, wherein the aryl group at the 8-position contains a substituent substituted-alkenyl group, are PDE4 inhibitors.
申请公布号 WO02069970(A1) 申请公布日期 2002.09.12
申请号 WO2001US48674 申请日期 2001.12.14
申请人 MERCK & CO., INC.;MERCK FROSST CANADA & CO.;VAILAYA, ANANT;CONLON, DAVID, A.;HO, GUO-JIE;MACDONALD, DWIGHT;PERRIER, HELENE;THIBERT, ROCH;KWONG, ELIZABETH;CLAS, SOPHIE-DOROTHEE 发明人 VAILAYA, ANANT;CONLON, DAVID, A.;HO, GUO-JIE;MACDONALD, DWIGHT;PERRIER, HELENE;THIBERT, ROCH;KWONG, ELIZABETH;CLAS, SOPHIE-DOROTHEE
分类号 A61K31/47;A61K31/4709;A61K45/00;A61P1/04;A61P7/00;A61P9/00;A61P9/10;A61P11/00;A61P11/02;A61P11/06;A61P11/14;A61P13/00;A61P13/12;A61P17/00;A61P17/04;A61P17/06;A61P19/02;A61P19/10;A61P21/00;A61P25/00;A61P25/04;A61P25/16;A61P25/24;A61P25/28;A61P27/02;A61P29/00;A61P31/04;A61P35/00;A61P37/06;A61P37/08;A61P43/00;C07D215/12;C07D215/14;C07D401/10;C07D413/10;C07D417/10;(IPC1-7):A61K31/47 主分类号 A61K31/47
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