发明名称 METHOD FOR THE PRODUCTION OF 4-(17ALPHA SUBSTITUTED 3-OXOESTRA-4,9-DIEN-11-YL)BENZALDEHYD-(1E OR 1Z)-OXIMES
摘要 The invention relates to a method for the production of 4-(17 substituted 3-oxoestra-4,9-dien-11 -yl)benzaldehyd-(1E or 1Z)-oximes of general formula (I), where R1 = H, C1-6 alkyl or a CnF2n+1 group; R2 = C1-4 alkyl, X = E- or Z-OH; and Y = O-C1-6 alkyl, S-C1-6 alkyl or O-CH2CnF2n+1, where n = 1, 2 or 3, which produces the target compounds of formula (I) with high yield and selectivity.
申请公布号 WO0238582(A3) 申请公布日期 2002.09.12
申请号 WO2001DE04218 申请日期 2001.11.09
申请人 JENAPHARM GMBH & CO. KG;SCHUBERT, GERD;RING, SVEN;ERHART, BERND 发明人 SCHUBERT, GERD;RING, SVEN;ERHART, BERND
分类号 C07J1/00;C07J21/00;C07J41/00;C07J71/00 主分类号 C07J1/00
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