发明名称 NITROGENOUS HETEROAROMATIC RING DERIVATIVE HAVING HIV INTEGRASE INHIBITORY ACTIVITY
摘要 A compound represented by the formula (I): (I) wherein ring A is a nitrogenous heteroaromatic ring; X is oxygen, sulfur, or NH; and R<A> is a group represented by the formula (II) (II) (wherein ring B is a nitrogenous heteroaromatic ring), etc. It has integrase inhibitory activity.
申请公布号 WO02070491(A1) 申请公布日期 2002.09.12
申请号 WO2002JP01779 申请日期 2002.02.27
申请人 SHIONOGI & CO., LTD.;FUJI, MASAHIRO 发明人 FUJI, MASAHIRO
分类号 A61P31/12;A61P31/18;A61P43/00;C07D235/24;C07D401/06;C07D403/06;C07D417/06;(IPC1-7):C07D235/12;C07D263/32;C07D277/24;C07D213/50;C07D239/26;C07D241/12;C07D263/56;C07D277/64;C07D239/74;C07D241/42;C07D471/04;C07D498/04;C07D513/04;C07D487/04;A61K31/418;A61K31/427;A61K31/443;A61K31/437;A61K31/472;A61K31/506;A61K31/501 主分类号 A61P31/12
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