发明名称 |
Process for water soluble azole compounds |
摘要 |
An improved process is provided for preparing water-soluble prodrugs of triazole antifungal compounds containing a secondary or tertiary hydroxyl group. More particularly, the improved process is directed toward preparation of water-soluble triazole antifungal compounds are provided having the general formulawherein A is the non-hydroxy portion of a triazole antifungal compound of the type containing a secondary or tertiary hydroxyl group and R and R1 are as defined in the specification.
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申请公布号 |
US6448401(B1) |
申请公布日期 |
2002.09.10 |
申请号 |
US20010982199 |
申请日期 |
2001.10.16 |
申请人 |
BRISTOL-MYERS SQUIBB COMPANY |
发明人 |
CHEN CHUNG-PIN;CONNOLLY TIMOTHY PAUL;KOLLA LAXMA REDDY;MATISKELLA JOHN D.;MUELLER RICHARD H.;PENDRI YADAGIRI;PETSCH DEJAH T. |
分类号 |
C07F9/6539;C07D249/08;C07D277/22;C07F9/6518;C07F9/6558;(IPC1-7):C07F9/02;C07F9/06 |
主分类号 |
C07F9/6539 |
代理机构 |
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