发明名称 |
STABLE RADIOIODINE CONJUGATES AND METHODS FOR THEIR SYNTHESIS |
摘要 |
Methods are described for conjugating radioiodinated peptides to non-metabolizable carbohydrates with improved yields and qualities of conjugates. Radioiodinated residualizing antibody conjugates comprising a carbohydrate-appended peptide are also provided. The instant radioiodinated residualizing antibody conjugates are particularly stable in vivo and are suitable for radioimmunodetection and radioimmunotherapy. |
申请公布号 |
WO0202150(A3) |
申请公布日期 |
2002.09.06 |
申请号 |
WO2001US20764 |
申请日期 |
2001.06.29 |
申请人 |
IMMUNOMEDICS, INC.;GOVINDAN, SERENGULAM, V. |
发明人 |
GOVINDAN, SERENGULAM, V. |
分类号 |
A61K51/04;A61K51/08;A61K51/10;C07H3/04;C07K1/107;G01N33/543 |
主分类号 |
A61K51/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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