| 摘要 |
2-Oxo-2,3-dihydroindole -3-carboxamides Title compds. (I) useful as anti-inflammatory agents (where X and Y are H, F, Cl or Br, 1-5C alkyl or alkoxy, CF3 or OCF3; R1 is H, CH2CF3 1-6C alkyl, 2-4C alkenyl or phenyl alkyl (1-3C alkyl); R2 is naphthyl or phenyl opt. substd. by one or two Cl, F, Br, 1-4C alkyl, 1-3C alkoxy or -alkylthio, CF3 or OCF3) are prepd. by reaction of a 2-oxo-2,3-dihydroindole with R2 NCO or with (Acyl)2 N-CONHR2 or by amidation of the 3-carboxylate.
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