发明名称 |
2-(2-Amino-1,6-dihydro-6-oxopurin-9-yl)methoxy-3-hydroxy-1-propanyl-L-valinate and its use, intermediate and pharmaceutical composition |
摘要 |
<p>2-(2-Amino-1,6-dihydro-6-oxopurin-9-yl)methoxy-3-hydroxy-1-propanyl-L-valin t nebo jeho farmaceuticky akceptovateln s l, ve form (R)- nebo (S)-diastereomeru nebo ve form sm s t chto dvou diastereomer . Pou it tohoto L-valin tu pro p° pravu farmaceutick²ch kompozic pro l en virov²ch a p° buzn²ch nemoc a tyto kompozice. Meziprodukt pro v²robu tohoto valin tu, vzorce II, kde P.sup.1.n. je vod k, nebo hydroxy-chr nic skupina a P.sup.2.n. je amino-chr nic skupina./</p> |
申请公布号 |
CZ290511(B6) |
申请公布日期 |
2002.08.14 |
申请号 |
CZ19950001939 |
申请日期 |
1995.07.27 |
申请人 |
F. HOFFMANN-LA ROCHE AG |
发明人 |
NESTOR JOHN J.;WOMBLE SCOTT W.;MAAG HANS |
分类号 |
C07D473/18;A61K31/198;A61K31/52;A61K31/522;A61P31/12;A61P31/22;A61P43/00;C07D473/00;(IPC1-7):C07D473/18 |
主分类号 |
C07D473/18 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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