发明名称 Pyrimidine-5-carboxamide derivatives
摘要 Pyrimidine-5-carboxamide derivatives represented by a general formula (I) or salts thereof[wherein each symbol has the following meaning;X: O, S, NR1, CO, NR1CO, CONR1, C=N-OR1 or a bond,Y: a lower alkylene group which may be substituted by OR1 or -NHR1, or a bond,Z: O, NR2 or a bond,A: H, or a lower alkyl which may have a substituent, a -CO-lower alkyl which may have a substituent, an aryl which may have a substituent, a heteroaryl which may have a substituent, a cycloalkyl which may have a substituent or a nitrogen-containing saturated heterocyclic group which may have a substituent,B: an aryl which may have a substituent or a heteroaryl group which may have a substituent,R1, R2: H, a lower alkyl or a -CO-lower alkyl group].
申请公布号 US6432963(B1) 申请公布日期 2002.08.13
申请号 US20000581595 申请日期 2000.06.15
申请人 YAMANOUCHI PHARMACEUTICAL CO., LTD. 发明人 HISAMICHI HIROYUKI;NAITO RYO;KAWAZOE SOUICHIROU;TOYOSHIMA AKIRA;TANABE KAZUHITO;NAKAI EIICHI;ICHIKAWA ATSUSHI;ORITA AKIKO;TAKEUCHI MAKOTO
分类号 A61P37/08;C07D239/38;C07D239/42;C07D239/46;C07D239/48;C07D239/56;C07D401/12;C07D403/12;C07D405/12;C07D409/12;C07D417/12;C07D521/00;(IPC1-7):C07D239/48;A61K31/505 主分类号 A61P37/08
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