发明名称 |
PIPERAZINE DERIVATIVES, THEIR PREPARATION AND THEIR USE FOR TREATING CENTRAL NERVOUS SYSTEM (CNS) DISORDERS |
摘要 |
Novel piperazine derivatives are provided having the formula (III) wherein R>1< is cyano, notro, trifluoromethyl or halogen, or pharmaceutically acceptable acid addition salts thereof, which are useful as 5-HT>1A< receptor antagonists. |
申请公布号 |
WO0244142(A3) |
申请公布日期 |
2002.08.08 |
申请号 |
WO2001US43160 |
申请日期 |
2001.11.27 |
申请人 |
WYETH |
发明人 |
CHILDERS, WAYNE, EVERETT;KELLY, MICHAEL, GERARD;ROSENZWEIG-LIPSON, SHARON, JOY |
分类号 |
A61K31/496;A61P1/14;A61P5/00;A61P9/00;A61P13/02;A61P15/10;A61P25/00;A61P25/06;A61P25/14;A61P25/16;A61P25/18;A61P25/20;A61P25/22;A61P25/24;A61P25/28;A61P25/30;A61P25/32;A61P25/34;A61P25/36;A61P43/00;C07B55/00;C07B57/00;C07D405/12 |
主分类号 |
A61K31/496 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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