发明名称 |
CAPROLACTAM DERIVATIVES AND USES THEREOF |
摘要 |
The invention involves derivatives of caprolactam of the formula (I) in which [A<1>], A<2> and R<1> have the meanings indicated in the description, their salts and their prodrugs. The invention also relates to the preparation of such compounds, synthetic intermediates, their use, and in particular, antagonists of the Src SH2 domain and inhibitors of bone resorption and pharmaceutical compounds containing such compounds.
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申请公布号 |
WO0168655(A3) |
申请公布日期 |
2002.08.01 |
申请号 |
WO2001US07935 |
申请日期 |
2001.03.12 |
申请人 |
ARIAD PHARMACEUTICALS, INC.;DEPREZ, PIERRE;LESUISSE, DOMINIQUE;BENARD, DIDIER |
发明人 |
DEPREZ, PIERRE;LESUISSE, DOMINIQUE;BENARD, DIDIER |
分类号 |
A61K38/00;C07F9/12;C07F9/40;C07F9/553;C07K5/06;C07K5/065;(IPC1-7):C07K5/065;C07K5/068;A61K38/05;A61K31/675;C07D223/12;C07C233/47 |
主分类号 |
A61K38/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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