发明名称 PROCESS FOR THE PREPARATION OF HETEROCYCLIC INDENE ANALOGS
摘要 The present invention is concerned with a novel process for the preparation of compounds of formula (I) wherein R<1>, R<2> and X are as defined in the specification, comprising cyclocarbonylation of a compound of formula (II) wherein R<1>, R<2>, R<3> and X are as defined in the specification, to produce a compound of formula (III) wherein R<1>, R<2>, R<4> and X are as defined in the specification, followed by saponification.
申请公布号 WO02059089(A2) 申请公布日期 2002.08.01
申请号 WO2002EP00583 申请日期 2002.01.22
申请人 F. HOFFMANN-LA ROCHE AG 发明人 SCALONE, MICHELANGELO;ZEIBIG, THOMAS
分类号 C07B61/00;C07D209/12;C07D209/88;C07D405/12 主分类号 C07B61/00
代理机构 代理人
主权项
地址