发明名称 THIAZOLE AND OXAZOLE DERIVATIVES AS ACTIVATORS OF HUMAN PEROXISOME PROLIFERATOR ACTIVATED RECEPTORS
摘要 The present invention provides a compound of formula (I) wherein R>1<-R>5<, R>25<, R>26<, Y and X>2< are defined as in claim 1. The compounds activate human peroxisome proliferator activated receptors (hPPARs) and are useful for the treatment of associated disorders such as cardiovascular disease and hypercholesteremia.
申请公布号 WO02059098(A1) 申请公布日期 2002.08.01
申请号 WO2001US51056 申请日期 2001.12.19
申请人 GLAXO GROUP LIMITED;BANKER, PIERETTE;CADILLA, RODOLFO;LAMBERT, MILLARD, HURST, III;RAFFERTY, STEPHEN, WILLIAM;STERNBACH, DANIEL, DAVID;SZNAIDMAN, MARCOS, LUIS 发明人 BANKER, PIERETTE;CADILLA, RODOLFO;LAMBERT, MILLARD, HURST, III;RAFFERTY, STEPHEN, WILLIAM;STERNBACH, DANIEL, DAVID;SZNAIDMAN, MARCOS, LUIS
分类号 C07D233/64;A61K31/426;A61K31/427;A61K31/496;A61K31/497;A61K31/506;A61P1/14;A61P3/04;A61P3/06;A61P3/10;A61P9/00;A61P9/04;A61P9/10;A61P25/00;A61P43/00;C07D263/32;C07D277/24;C07D277/26;C07D277/28;C07D417/06;C07D417/10;C07D417/12;C07F7/12;(IPC1-7):C07D277/24;A61K31/42;A61K31/425 主分类号 C07D233/64
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