发明名称 |
OPTICALLY ACTIVE ENANTIOMER OF 5-[3-(EXO-BICYCLO[2.2.1]HEPT-2-YL-OXY)-4-METHOXY-PHENYL]-3,4,5,6-TETRAHYDROPYRIMIDIN-2(1H)-ONE AND INTERMEDIERS |
摘要 |
Process for the pancreatic lipase mediated transesterification method for the optical resolution of endo-norborneol; derived optically active 5-(3-(exo-bicyclo[2.2.1]hept-2-yloxy)-4-methoxyphenyl)-3,4,5,6-tetrahy dropyrimid in-2(1H)-ones; and stepwise process and intermediates therefor. |
申请公布号 |
HU220962(B1) |
申请公布日期 |
2002.07.29 |
申请号 |
HU19980002988 |
申请日期 |
1989.11.13 |
申请人 |
PFIZER INC. |
发明人 |
SACCOMANO NICHOLAS A. |
分类号 |
C07D239/20;A61K31/505;A61K31/513;A61P11/00;A61P11/06;A61P11/08;A61P17/00;C07C35/22;C07C35/29;C07C45/71;C07C47/575;C07C225/34;C07C233/00;C07C233/11;C07C233/29;C07C235/34;C07C255/04;C07C255/32;C07C255/35;C07C255/37;C07D239/10;C07D239/14;C12P7/02;C12P41/00 |
主分类号 |
C07D239/20 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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