发明名称 NOVEL COMPOUNDS AND COMPOSITIONS AS CATHEPSIN INHIBITORS
摘要 The present invention relates to novel selective cathepsin S inhibitors, the pharmaceutically acceptable salts and N-oxides thereof, their uses as therapeutic agents and the methods of their making
申请公布号 WO02051983(A2) 申请公布日期 2002.07.04
申请号 WO2001US50680 申请日期 2001.12.24
申请人 CELERA, AN APPLERA CORPORATION BUSINESS;GRAUPE, MICHAEL;PATTERSON, JOHN;PICKETT, STEPHEN, D.;LINK, JOHN;LI, JIAYAO;ALDOUS, DAVID;THURAIRATNAM, SUKANTHINI;TIMM, ANDREAS;HALLEY, FRANK;LAI, JUSTINE 发明人 GRAUPE, MICHAEL;PATTERSON, JOHN;PICKETT, STEPHEN, D.;LINK, JOHN;LI, JIAYAO;ALDOUS, DAVID;THURAIRATNAM, SUKANTHINI;TIMM, ANDREAS;HALLEY, FRANK;LAI, JUSTINE
分类号 C07D295/18;A61K31/165;A61K31/277;A61K31/423;A61K31/4245;A61K31/425;A61K31/437;A61K31/454;A61K31/5375;A61K31/5377;A61K31/55;A61P3/10;A61P9/10;A61P11/00;A61P11/06;A61P17/00;A61P19/02;A61P21/04;A61P25/00;A61P25/28;A61P29/00;A61P37/02;A61P37/08;A61P43/00;C07C317/44;C07C317/50;C07C323/60;C07D205/08;C07D205/085;C07D207/24;C07D207/26;C07D207/273;C07D213/40;C07D223/10;C07D223/12;C07D263/06;C07D263/32;C07D263/56;C07D271/06;C07D271/10;C07D277/26;C07D277/64;C07D285/08;C07D295/185;C07D413/04;C07D413/12;C07D498/04 主分类号 C07D295/18
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