发明名称 |
BRIDGED NICOTINE COMPOUNDS FOR USE IN THE TREATMENT OF CNS PATHOLOGIES |
摘要 |
Pharmaceutical compounds commprising bridged nicotine analogs of N-octylnicotinium iodide (NONI) having selective antagonist properties at alpha 3 beta 2-containing nicotinic receptor subtypes, and compositions containing these compounds. The compounds and compositions are used to treat central nervous system pathologies.
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申请公布号 |
WO0217922(A8) |
申请公布日期 |
2002.07.04 |
申请号 |
WO2001US26876 |
申请日期 |
2001.08.30 |
申请人 |
UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION |
发明人 |
CROOKS, PETER;DWOSKIN, LINDA;XU, RUI;GRINEVICH, VLADIMIR |
分类号 |
C07D471/04;(IPC1-7):A61K31/474;C07D471/02 |
主分类号 |
C07D471/04 |
代理机构 |
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