发明名称 |
AMIDE DERIVATIVES OF ANTIBIOTIC A 40926 |
摘要 |
The present invention is directed to novel antibiotic A 40926 derivatives characterized by having a carboxy, (C1-C4)alkoxy- carbonyl, aminocarbonyl, (C1-C4)alkylaminocarbonyl, di(C1- C4)alkylaminocarbonyl or hydroxymethyl substituent on the N-acylaminoglucuronyl moiety and a hydroxy or a polyamine substituent in position 63 of the molecule. The compounds of the invention show high in vitro activity against glycopeptide resistant Enterococci and Staphylococci.
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申请公布号 |
CA2109601(C) |
申请公布日期 |
2002.07.02 |
申请号 |
CA19922109601 |
申请日期 |
1992.07.14 |
申请人 |
GRUPPO LEPETIT S.P.A. |
发明人 |
MALABARBA, ADRIANO;CIABATTI, ROMEO;PANZONE, GIANBATTISTA;MARAZZI, ALESSANDRA M. |
分类号 |
A61K38/00;A61K31/7048;A61K31/7052;A61K38/04;A61P31/04;C07H17/08;C07K1/113;C07K9/00;C07K14/195;C07K14/41;(IPC1-7):C07K9/00;A61K38/14;C07K1/00 |
主分类号 |
A61K38/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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