发明名称 |
PYRAZOLO[3,4-C]PYRIDINES AS GSK-3 INHIBITORS |
摘要 |
A compound of formula (I) or a derivative thereof, wherein R<1> is unsubstituted or substituted alkyl, unsubstituted or substituted cycloalkyl, unsubstituted or substituted alkenyl, unsubstituted or substituted cycloalkenyl, unsubstituted or substituted aryl, aralkyl wherein the aryl and the alkyl moieties may each independently be unsubstituted or substituted, aralkenyl wherein the aryl and alkenyl moieties may each independently be unsubstituted or substituted, unsubstituted or substituted heterocyclyl, or heterocyclyalkyl wherein the heterocyclyl and the alkyl moieties may each independently be unsubstituted or substituted; and R<2> is unsubstituted or substituted aryl or unsubstituted or substituted heteroaryl, a process for preparing such compounds, a pharmaceutical composition comprising such compounds and the use of such compounds and composition in medicine.
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申请公布号 |
WO0250073(A1) |
申请公布日期 |
2002.06.27 |
申请号 |
WO2001GB05663 |
申请日期 |
2001.12.19 |
申请人 |
SMITHKLINE BEECHAM P.L.C.;RAWLINGS, DEREK, ANTHONY;WITHERINGTON, JASON |
发明人 |
RAWLINGS, DEREK, ANTHONY;WITHERINGTON, JASON |
分类号 |
A61K31/437;A61P3/04;A61P3/10;A61P7/00;A61P7/04;A61P9/10;A61P9/12;A61P15/08;A61P17/02;A61P17/14;A61P21/04;A61P25/00;A61P25/14;A61P25/16;A61P25/18;A61P25/28;A61P31/00;A61P31/18;A61P35/00;A61P37/00;A61P43/00;C07D471/04;(IPC1-7):C07D471/04 |
主分类号 |
A61K31/437 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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