发明名称 |
SUBSTITUTED BENZOINDOLES AS SPLA2 INHIBITORS |
摘要 |
A novel class of benz[f]indole compounds see structure (I) is disclosed together with the use of such compounds for inhibiting sPLA2 mediated releas e of fatty acids for treatment of inflammatory diseases such as septic shock.< /SDOAB>
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申请公布号 |
CA2431023(A1) |
申请公布日期 |
2002.06.27 |
申请号 |
CA20012431023 |
申请日期 |
2001.12.06 |
申请人 |
ELI LILLY AND COMPANY |
发明人 |
KINNICK, MICHAEL DEAN;LIN, HO-SHEN;SMITH, EDWARD C. R.;SAWYER, JASON SCOTT;MORIN, JOHN MICHAEL JUNIOR;SALL, DANIEL JON;BEIGHT, DOUGLAS WADE;RICHETT, MICHAEL ENRICO |
分类号 |
A61K31/403;A61P1/04;A61P3/00;A61P3/12;A61P5/06;A61P5/18;A61P7/00;A61P7/04;A61P9/00;A61P11/00;A61P11/02;A61P11/06;A61P13/12;A61P17/02;A61P17/06;A61P19/02;A61P19/04;A61P19/06;A61P19/08;A61P21/00;A61P29/00;A61P31/04;A61P31/06;A61P31/10;A61P31/12;A61P35/00;A61P37/08;A61P43/00;C07D209/60;(IPC1-7):C07D209/00;A61K31/40 |
主分类号 |
A61K31/403 |
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