发明名称 |
SUBSTITUTED N-PIPERIDINO-PYRAZOLE-3-CARBOXAMIDE |
摘要 |
<p>N-piperidino-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4- methylpyrazole-3-carboxamide of the formula: its pharmaceutically acceptable salts and their solvates, are potent antagonists of the central cannabinoid receptors. They are prepared by reaction of a functional derivative of 5-(4- chlorophenyl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3- carboxylic acid with 1-aminopiperidine and, optionally, formation of a salt.</p> |
申请公布号 |
CA2136893(C) |
申请公布日期 |
2002.06.25 |
申请号 |
CA19942136893 |
申请日期 |
1994.11.29 |
申请人 |
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发明人 |
BARTH, FRANCIS;CASELLAS, PIERRE;CONGY, CHRISTIAN;MARTINEZ, SERGE;RINALDI, MURIELLE;ANN-ARCHARD, GILLES |
分类号 |
C07D401/12;A61K31/415;A61K31/4465;A61K31/4523;A61K31/454;A61P1/08;A61P1/14;A61P7/02;A61P25/00;A61P25/04;A61P25/06;A61P25/08;A61P25/14;A61P25/16;A61P25/18;A61P25/20;A61P25/22;A61P25/28;A61P29/00;A61P43/00;C07D231/14;C07D231/40;(IPC1-7):C07D401/12;A61K31/445 |
主分类号 |
C07D401/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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