发明名称 A PROCESS FOR THE PREPARATION OF N,N'-SUBSTITUTED 5-AMINO-1,3-BENZENEDICARBOXAMIDES
摘要 The invention relates to a process for the preparation of a compound of formula (I), wherein R represents a 2,3-dihydroxy-1-propyl or a 1,3-dihydroxy-2-propyl radical, via direct amidation of a dialkyl ester of 5-amino-1,3-benzenedicarboxylic acid of formula (V), wherein R1 represents a straight or branched (C1-C4)-alkyl group, with at least the stoichiometric amount of an amine of formula H2NR.
申请公布号 WO0244125(A1) 申请公布日期 2002.06.06
申请号 WO2001EP13879 申请日期 2001.11.28
申请人 BRACCO IMAGING S.P.A.;ANELLI, PIER, LUCIO;BROCCHETTA, MARINO;LUX, GIOVANNA;CAPPELLETTI, ENRICO 发明人 ANELLI, PIER, LUCIO;BROCCHETTA, MARINO;LUX, GIOVANNA;CAPPELLETTI, ENRICO
分类号 C07C227/04;C07C227/18;C07C231/02;C07C231/12;C07C231/14;C07C237/32;C07C237/42;(IPC1-7):C07C231/02 主分类号 C07C227/04
代理机构 代理人
主权项
地址