发明名称 |
A PROCESS FOR THE PREPARATION OF N,N'-SUBSTITUTED 5-AMINO-1,3-BENZENEDICARBOXAMIDES |
摘要 |
The invention relates to a process for the preparation of a compound of formula (I), wherein R represents a 2,3-dihydroxy-1-propyl or a 1,3-dihydroxy-2-propyl radical, via direct amidation of a dialkyl ester of 5-amino-1,3-benzenedicarboxylic acid of formula (V), wherein R1 represents a straight or branched (C1-C4)-alkyl group, with at least the stoichiometric amount of an amine of formula H2NR.
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申请公布号 |
WO0244125(A1) |
申请公布日期 |
2002.06.06 |
申请号 |
WO2001EP13879 |
申请日期 |
2001.11.28 |
申请人 |
BRACCO IMAGING S.P.A.;ANELLI, PIER, LUCIO;BROCCHETTA, MARINO;LUX, GIOVANNA;CAPPELLETTI, ENRICO |
发明人 |
ANELLI, PIER, LUCIO;BROCCHETTA, MARINO;LUX, GIOVANNA;CAPPELLETTI, ENRICO |
分类号 |
C07C227/04;C07C227/18;C07C231/02;C07C231/12;C07C231/14;C07C237/32;C07C237/42;(IPC1-7):C07C231/02 |
主分类号 |
C07C227/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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