发明名称 NEW BENZENESULPHONAMIDE COMPOUNDS, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.
摘要 Compound of formula (I): wherein: n is from 1 to 3, and m is from 0 to 6, Ra represents hydroxy, alkoxy, aryloxy or arylalkyloxy, R1 and R2 represent independently hydrogen, halogen, alkyl, alkoxy, hydroxy or perhaloalkyl, R3 represents hydrogen, or alkyl, arylalkyl, cycloalkylalkyl, aryl or cycloalkyl, T1 represents alkylene, O-alkylene, alkylene-O- or (C1-C3)alkylene-O- (C1-C3)alkylene, G represents G1- or G1-T2-A-, wherein: A represents aryl, T2 represents a bond or alkylene, -O-alkylene, alkylene-O- or (C1-C3)-alkylene-O-(C1-C3)alkylene, G1 represents -NR4R5, or G1 represents heterocycloalkyl a formula having from 5 to 7 ring members wherein Y represents a nitrogen atom, oxygen or CH and R4, R5 and R6 are as defined in the description, and medicinal products containing the same are useful as TXA2 receptor antagonist and 5-HT2 receptor antagonist.
申请公布号 MXPA01000363(A) 申请公布日期 2002.06.04
申请号 MX2001PA00363 申请日期 2001.01.10
申请人 LES LABORATOIRES SERVIER. 发明人 GILBERT LAVIELLE
分类号 C07D295/08;A61K31/40;A61K31/4427;A61K31/4433;A61K31/445;A61K31/4535;A61K31/454;A61K31/495;A61K31/496;A61P7/00;A61P7/02;A61P9/08;A61P9/10;A61P11/00;A61P11/06;A61P11/08;A61P25/06;A61P43/00;C07D207/08;C07D211/14;C07D211/18;C07D211/22;C07D211/32;C07D211/70;C07D295/096;C07D295/18;C07D295/192;C07D401/04;C07D409/04;C07D413/04;C07D417/04;(IPC1-7):A61K31/445;C07D241/04;C07D295/00 主分类号 C07D295/08
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