发明名称 |
Paclitaxel Prodrogen, Verfahren zur Herstellung und ihre Verwendung zur selektiven Chemotherapie |
摘要 |
A paclitaxel prodrug has a paclitaxel portion coupled to a cleavable N-(aliphatic or aromatic)-O-glycosyl carbamate spacer group, and can be administered orally, topically or by injection to provide an anti-tumor effect, the prodrug being activated by a hydrolizing enzyme, an endogeneous enzyme or an exogeneous enzyme. |
申请公布号 |
DE69620727(D1) |
申请公布日期 |
2002.05.23 |
申请号 |
DE1996620727 |
申请日期 |
1996.12.17 |
申请人 |
PHARMACHEMIE B.V., HAARLEM |
发明人 |
DE BONT, HENDRICUS BARTHELOMEAS ANDREAS;HAISMA, HIDDE JACOB;LEENDERS, RUBEN GERADUS GEORGE;DE VOS, DICK;SCHEEREN, JOHAN WILHELM |
分类号 |
C07D305/14;A61K31/335;A61K31/337;A61K31/70;A61K31/7024;A61K38/46;A61K39/395;A61K47/48;A61P35/00;A61P43/00;C07C263/12;C07H13/12;(IPC1-7):C07H13/10;C07C265/04;C07C265/12 |
主分类号 |
C07D305/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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