| 发明名称 |
PYRAZOLECARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
| 摘要 |
<p>N-Piperidino-5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-ethylpyrazole -3-carboxamide and its salts and solvates are powerful antagonists of the CB1 cannabinoid receptors. They are prepared by reacting a functional derivative of 5-(4-bromophenyl)-1-(2,4-dichlorophenyl) -4-ethylpyrazole-3-carboxylic acid with 1-aminopiperidine, optionally followed by salification.</p> |
| 申请公布号 |
IL144198(D0) |
申请公布日期 |
2002.05.23 |
| 申请号 |
IL20000144198 |
申请日期 |
2000.01.28 |
| 申请人 |
SANOFI-SYNTHELABO |
发明人 |
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| 分类号 |
A61K31/415;A61K31/454;A61P3/00;A61P3/04;A61P25/00;A61P25/18;A61P25/28;A61P25/32;A61P25/34;A61P43/00;C07C69/738;C07C251/80;C07D231/14;(IPC1-7):C07D |
主分类号 |
A61K31/415 |
| 代理机构 |
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代理人 |
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| 主权项 |
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| 地址 |
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