发明名称 Thrombin inhibitors
摘要 This application relates to novel compounds of formula I (and their pharmaceutically acceptable salts), as defined herein, processes and intermediates for their preparation, pharmaceutical formulations comprising the novel compounds of formula I, and the use of defined compounds of formula I as thrombin inhibitors.
申请公布号 US6391901(B1) 申请公布日期 2002.05.21
申请号 US20000423148 申请日期 2000.01.21
申请人 ELI LILLY AND COMPANY 发明人 CHIRGADZE NICKOLAY Y;DENNEY MICHAEL L;FISHER MATTHEW J;FOGLESONG ROBERT J;HARPER RICHARD W;JOHNSON MARY G;LIN HO-SHEN;LYNCH MICHAEL P;MCCOWAN JEFFERSON R;MILLER SHAWN C;PALKOWITZ ALAN D;RICHETT MICHAEL E;SALL DANIEL J;SMITH GERALD F;TAKEUCHI KUMIKO;ZHANG MINSHENG
分类号 C07D409/14;A61K31/4025;A61K31/4155;A61K31/4166;A61K31/4178;A61K31/422;A61K31/427;A61K31/4439;A61K31/454;A61K31/5377;A61P7/02;C07D333/56;C07D333/58;C07D409/12;C07D413/12;C07D413/14;C07D417/12;C07D417/14;(IPC1-7):A61K31/402;A61K31/417;A61K31/381;C07D333/52 主分类号 C07D409/14
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