发明名称 |
PROCESS FOR THE PREPARATION OF NON-STEROIDAL GLUCOCORTICOID RECEPTOR MODULATORS |
摘要 |
PURPOSE: Provided is a process for preparing a compound of the formula(1) useful as a non-steroidal glucocorticoid receptor modulator. CONSTITUTION: The process for preparing a compound of the formula(1) characteristically comprises reacting a compound of the formula(2) with an amide in the presence of 1,1'-carbonyldiimazole.
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申请公布号 |
KR20020033075(A) |
申请公布日期 |
2002.05.04 |
申请号 |
KR20010066290 |
申请日期 |
2001.10.26 |
申请人 |
PFIZER PRODUCTS INC. |
发明人 |
MURRY JERRY ANTHONY;WHITE TIMOTHY DONALD |
分类号 |
A61K31/44;A61P5/44;A61P5/46;A61P43/00;C07B61/00;C07C35/42;C07C41/26;C07C43/188;C07C43/192;C07C43/196;C07C49/747;C07C51/08;C07C63/70;C07C65/17;C07C253/30;C07C255/26;C07C255/53;C07C255/54;C07C255/56;C07C269/00;C07C271/52;C07D213/38;C07D213/40;(IPC1-7):C07D213/40 |
主分类号 |
A61K31/44 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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