发明名称 |
DRUG COMPOSITION COMPRISING DIPEPTYDYL ALDEHYDE DERIVATIVE |
摘要 |
A drug composition which comprises a compound represented by the general formula (I), wherein R<1> represents an alkyl group having 1 to 4 carbon atoms or represents an aryl group having 6 to 10 carbon atoms optionally having a substituent, R<2> and R<3> may be the same or different and each represent hydrogen or an alkyl group having 1 to 4 carbon atoms or R<2> and R<3> may together form a ring having 3 to 7 carbon atoms, and R<4> represents an aryl group, a cycloalkyl group or a lower alkyl group optionally substituted with an aromatic heterocyclic residue, or a pharmaceutically acceptable salt of the compound, and a lipid. The drug composition is improved in stability, absobability and the transfer to a target tissue over a conventional composition containing no lipid added.
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申请公布号 |
WO0234252(A1) |
申请公布日期 |
2002.05.02 |
申请号 |
WO2001JP08514 |
申请日期 |
2001.09.27 |
申请人 |
SENJU PHARMACEUTICAL CO., LTD.;INOUE, JUN;YAMAGUCHI, MASAZUMI |
发明人 |
INOUE, JUN;YAMAGUCHI, MASAZUMI |
分类号 |
A61K9/00;A61K9/127;A61K9/48;A61K31/18;A61K31/404;A61K47/02;A61K47/24;A61K47/28;A61K47/48;A61P9/10;A61P19/10;A61P25/00;A61P25/28;A61P27/02;A61P27/06;A61P37/02;(IPC1-7):A61K31/18 |
主分类号 |
A61K9/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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