PROCESS FOR PREPARATION OF INTEGRIN RECEPTOR ANTAGONIST INTERMEDIATES
摘要
A novel process is provided for the preparation of chiral intermediates usef ul in the asymmetric syntheses of .alpha.v.beta.3 integrin receptor antagonists . Also provided are the enantiomerically enriched intermediates that are obtained from the process.
申请公布号
CA2424304(A1)
申请公布日期
2002.04.11
申请号
CA20012424304
申请日期
2001.10.01
申请人
MERCK & CO., INC.
发明人
MCWILLIAMS, JAMES CHRISTOPHER;WATERS, MARJORIE SEE;SAGER, JESS W.;HUMPHREY, GUY R.;ENG, KAN K.;BUCK, ELIZABETH;MALIGRES, PETER E.