发明名称 |
GLUCOPYRANOSYLOXYBENZYLBENZENE DERIVATIVES AND MEDICINAL COMPOSITIONS CONTAINING THE SAME |
摘要 |
Glucopyranosyloxybenzylbenzene derivatives represented by the following general formula (I) which have an improved oral absorbability, exert an excellent effect of inhibiting human SGLT2 activity <i>in vivo</i> and, therefore, are useful as preventives or remedies for diseases caused by hyperglycemia such as diabetes, complication of diabetes and obesity wherein P represents a group constituting a prodrug; and R represents lower alkyl, lower alkoxy, lower alkylthio, lower alkoxy lower alkyl, lower alkoxy lower alkoxy or lower alkoxy lower alkylthio.
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申请公布号 |
WO0228872(A1) |
申请公布日期 |
2002.04.11 |
申请号 |
WO2001JP08239 |
申请日期 |
2001.09.21 |
申请人 |
KISSEI PHARMACEUTICAL CO., LTD.;FUJIKURA, HIDEKI;FUSHIMI, NOBUHIKO;NISHIMURA, TOSHIHIRO;TATANI, KAZUYA;ISAJI, MASAYUKI |
发明人 |
FUJIKURA, HIDEKI;FUSHIMI, NOBUHIKO;NISHIMURA, TOSHIHIRO;TATANI, KAZUYA;ISAJI, MASAYUKI |
分类号 |
A61K31/7034;A61P3/04;A61P3/10;A61P43/00;C07H15/203;(IPC1-7):C07H15/203;A61K31/703 |
主分类号 |
A61K31/7034 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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