| 发明名称 |
STEREOSELECTIVE PROCESS FOR PREPARING CYCLOHEXYL AMINE DERIVATIVES |
| 摘要 |
A process for preparing (1R,3S)-3-(9-chloro-3-methyl-4-oxo-5H-(isoxazoloquinolin-5-yl))cyclohe xanecarboxylic acid and esters thereof, as represented by formulas II and III, wherein R is a lower alkyl groups, and A and B are N or O, provided that when A is N, B is O, or when A is O, B is N: Formula (III) and Formula (II).
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| 申请公布号 |
WO0224705(A1) |
申请公布日期 |
2002.03.28 |
| 申请号 |
WO2001US26023 |
申请日期 |
2001.09.13 |
| 申请人 |
ELI LILLY AND COMPANY;BARNETT, CHARLES, JACKSON;GU, RUI LIN;KOBIERSKI, MICHAEL, EDWARD |
发明人 |
BARNETT, CHARLES, JACKSON;GU, RUI LIN;KOBIERSKI, MICHAEL, EDWARD |
| 分类号 |
A61K31/4745;A61P35/00;A61P43/00;C07B53/00;C07D498/04;(IPC1-7):C07D498/04 |
主分类号 |
A61K31/4745 |
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