发明名称 NOVEL PYRIMIDINE DERIVATIVE AND NOVEL PYRIDINE DERIVATIVE
摘要 The achiral pyrimidine derivative and pyridine derivative respectively represented by the formulae or analogues of these. They have selective N-type calcium channel inhibitory activity, and showed analgesic activity upon oral administration. They are useful not only as therapeutic agents for pains but as ones for various diseases in which N-type calcium channels participate.
申请公布号 WO0222588(A1) 申请公布日期 2002.03.21
申请号 WO2001JP07841 申请日期 2001.09.10
申请人 AJINOMOTO CO.,INC.;OHNO, SEIJI;OTANI, KAYO;NIWA, SEIJI;IWAYAMA, SATOSHI;TAKAHARA, AKIRA;KOGANEI, HAJIME;ONO, YUKITSUGU;FUJITA, SHINICHI;TAKEDA, TOMOKO;HAGIHARA, MASAKO;OKAJIMA, AKIKO 发明人 OHNO, SEIJI;OTANI, KAYO;NIWA, SEIJI;IWAYAMA, SATOSHI;TAKAHARA, AKIRA;KOGANEI, HAJIME;ONO, YUKITSUGU;FUJITA, SHINICHI;TAKEDA, TOMOKO;HAGIHARA, MASAKO;OKAJIMA, AKIKO
分类号 A61K31/455;A61K31/496;A61K31/505;A61K31/506;A61K31/5377;A61K31/55;A61K31/551;A61P1/04;A61P9/10;A61P11/06;A61P25/00;A61P25/04;A61P25/06;A61P25/16;A61P25/28;A61P25/30;A61P43/00;C07D213/80;C07D213/82;C07D239/28;C07D239/34;C07D239/38;C07D239/42;C07D401/04;C07D403/04;C07D409/04;C07D417/04;(IPC1-7):C07D239/38;C07D239/08;C07D401/14;C07D401/06;C07D401/12;A61K31/537 主分类号 A61K31/455
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