发明名称 COMBRETASTATIN A-4 PHOSPHATE PRODRUG SALTS WITH NITROGEN-CONTAINING COMPOUNDS
摘要 Provided herein are novel and useful combretastatin A-4 prodrug salts that increase the solubility of combretastatin A-4, readily regenerate combretastatin A-4<i> in vivo </i>under normal physiological conditions, and which produce physiologically tolerable products as a result of the regeneration of combretastatin A-4.
申请公布号 WO0222626(A1) 申请公布日期 2002.03.21
申请号 WO2001US28401 申请日期 2001.09.12
申请人 BRISTOL-MYERS SQUIBB COMPANY;VENIT, JOHN, J.;DALI, MANDAR, V.;DALI, MANISHA, M.;HUANG, YANDE;DAHLHEIM, CHARLES, E.;TEJWANI, RAVINDRA, W. 发明人 VENIT, JOHN, J.;DALI, MANDAR, V.;DALI, MANISHA, M.;HUANG, YANDE;DAHLHEIM, CHARLES, E.;TEJWANI, RAVINDRA, W.
分类号 A61P35/00;C07C211/14;C07C215/10;C07C215/12;C07C229/08;C07C229/26;C07C279/14;C07D233/54;C07D233/61;C07F9/12;(IPC1-7):C07F9/12;C07D209/20;A61K31/66 主分类号 A61P35/00
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