发明名称 Novel synthesis of piperazine ring
摘要 A novel process for preparing a compound of the formula I: wherein R1 denotes substituted or unsubstituted alkyl, alkoxy, aryl, aryloxy or arylalkoxy; R2 denotes substituted or unsubstituted alkyl, alkoxy, aryl, aryloxy, arylalkoxy, tosyl, formyl, acetyl or amine; and R3 denotes substituted or unsubstituted alkyl, alkoxy, aryl, aryloxy or arylalkoxy is disclosed. These compounds are useful in the synthesis of the antidepressant mirtazapine and other tetracyclic compounds.
申请公布号 US2002035256(A1) 申请公布日期 2002.03.21
申请号 US20010939406 申请日期 2001.08.24
申请人 DOLITZKY BEN-ZION 发明人 DOLITZKY BEN-ZION
分类号 C07D241/04;C07D471/14;(IPC1-7):C07D241/04;C07D295/00 主分类号 C07D241/04
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